{"id":13366,"date":"2024-05-13T12:00:00","date_gmt":"2024-05-13T12:00:00","guid":{"rendered":"https:\/\/www.africa-press.net\/sao-tome-e-principe\/politique\/depression-la-piste-dun-traitement-aux-toxines-hallucinogenes-de-crapaud"},"modified":"2024-05-14T23:41:33","modified_gmt":"2024-05-14T23:41:33","slug":"depression-la-piste-dun-traitement-aux-toxines-hallucinogenes-de-crapaud","status":"publish","type":"post","link":"https:\/\/www.africa-press.net\/sao-tome-e-principe\/toutes-les-actualites\/depression-la-piste-dun-traitement-aux-toxines-hallucinogenes-de-crapaud","title":{"rendered":"D\u00e9pression : la piste d\u2019un traitement aux toxines hallucinog\u00e8nes de crapaud"},"content":{"rendered":"<p><span style=\"color: #ff6600\"><strong>Africa-Press &#8211; S\u00e3o Tom\u00e9 e Pr\u00edncipe. <\/strong><\/span>Un psyche\u0301de\u0301lique issu du venin d\u2019un crapaud toxique pourrait e\u0302tre un traitement contre la de\u0301pression et l\u2019anxie\u0301te\u0301. Ce n\u2019est pas la premie\u0300re fois que la recherche s\u2019inte\u0301resse aux possibilite\u0301s qu\u2019offrent les psyche\u0301de\u0301liques dans le traitement de maladies mentales. Pour le moment, la majorite\u0301 des travaux portait sur un re\u0301cepteur a\u0300 la se\u0301rotonine (5-HT2A). Mais ces nouveaux re\u0301sultats, publie\u0301s dans Nature, se concentrent sur une nouvelle cible.<\/p>\n<p><b>Du poison au traitement the\u0301rapeutique<\/b><\/p>\n<p>La se\u0301rotonine est une mole\u0301cule qui agi\u0302t comme un neurotransmetteur dans le cerveau. Elle influe sur l\u2019humeur et, lorsqu\u2019elle est a\u0300 un taux e\u0301quilibre\u0301, est associe\u0301e a\u0300 l\u2019e\u0301tat de bonheur. La se\u0301rotonine est aussi la cible des antide\u0301presseurs dans le traitement de troubles psychiatriques, comme l\u2019anxie\u0301te\u0301 ou la de\u0301pression.<\/p>\n<p>Appele\u0301s \u201cinhibiteurs se\u0301lectifs de la recapture de la se\u0301rotonine\u201d, ces me\u0301dicaments ont pour but d\u2019augmenter le niveau de se\u0301rotonine dans le cerveau. Ils font en sorte que la se\u0301rotonine reste plus longtemps dans la synapse, a\u0300 la jointure entre deux neurones. Les re\u0301cepteurs de la se\u0301rotonine sont alors plus stimule\u0301s.<\/p>\n<p>Cette fois, l\u2019e\u0301quipe de l\u2019e\u0301cole de me\u0301decine de Mount Sinai a voulu trouver une substance capable de mieux stimuler ces re\u0301cepteurs. Elle s\u2019est pour cela inte\u0301resse\u0301e au crapaud Incilius alvarius.<\/p>\n<p>Surnomme\u0301 crapaud de la Colorado River (ou Colorado River Toad en anglais), on le retrouve aux E\u0301tats-Unis dans l\u2019extre\u0302me Sud-Est de la Californie, dans le Sud de l\u2019Arizona et dans l\u2019extre\u0302me Sud-Ouest du Nouveau-Mexique. Lorsqu\u2019il se sent en danger, ce crapaud toxique se\u0301cre\u0300te un poison associe\u0301 a\u0300 des expe\u0301riences psyche\u0301de\u0301liques intenses.<\/p>\n<p>L\u2019hallucinoge\u0300ne 5-MeO-DMT qu\u2019il produit interagit avec un re\u0301cepteur a\u0300 la se\u0301rotonine appele\u0301 5-HT1A. Apre\u0300s avoir examine\u0301 sa structure et modifie\u0301 certains sites spe\u0301cifiques, l\u2019e\u0301quipe a voulu e\u0301valuer le potentiel the\u0301rapeutique de cet agent dans le cadre de la de\u0301pression.<\/p>\n<p><b>Droit au but<\/b><\/p>\n<p>A ce stade de la recherche, l\u2019essai clinique n\u2019a pas e\u0301te\u0301 mene\u0301 sur l\u2019humain mais sur la souris. Sur une souris mode\u0301lisant la de\u0301pression, le nouveau compose\u0301 a montre\u0301 les me\u0302mes effets qu\u2019un traitement au LSD et qu\u2019un traitement a\u0300 base d\u2019antagonistes 5-HT1A de\u0301ja\u0300 identifie\u0301s. Mais, diffe\u0301rence notable, la mole\u0301cule s\u2019est montre\u0301e bien meilleure au moment d\u2019atteindre son but dans le cerveau.<\/p>\n<p>Compare\u0301 a\u0300 la cible 5-HT12, sur laquelle portent de\u0301ja\u0300 de nombreux travaux, le compose\u0301 s\u2019est montre\u0301 800 fois plus se\u0301lectif sur 5-HT1A. Cela signifie qu\u2019il parvenait a\u0300 toucher 800 fois mieux cette cible et qu\u2019elle pourrait e\u0302tre une cible the\u0301rapeutique potentielle. Surtout, aucun effet hallucinoge\u0300ne n\u2019a e\u0301te\u0301 rapporte\u0301, ce qui renforce son statut de possible candidat pour un traitement sur l\u2019humain.<\/p>\n<p>Gra\u0302ce a\u0300 ces travaux, les chercheurs espe\u0300rent re\u0301ussir a\u0300 dentifier quels psyche\u0301de\u0301liques parviennent le mieux a\u0300 moduler les re\u0301cepteurs dans le cerveau des mammife\u0300res. Cette nouvelle cible prometteuse pourrait faire l\u2019objet d\u2019une nouvelle classe de me\u0301dicaments destine\u0301s aux troubles neuropsychiatriques. Il faudra, en attendant, re\u0301ussir a\u0300 de\u0301montrer que ces premiers re\u0301sultats encourageants s\u2019appliquent aussi aux humains.<\/p>\n<p>Ce n\u2019est pas la premie\u0300re fois qu\u2019une substance hallucinoge\u0300ne est e\u0301tudie\u0301e pour traiter les troubles de\u0301pressifs. Re\u0301cemment, de nombreuses recherches ont porte\u0301 sur l\u2019apport des drogues psyche\u0301de\u0301liques comme le LSD.<\/p>\n<p>Le principe actif des champignons hallucinoge\u0300nes, la psilocybine, est e\u0301galement e\u0301tudie\u0301. Si ces expe\u0301riences ont montre\u0301 des re\u0301sultats inte\u0301ressants, elles ont e\u0301te\u0301 re\u0301alise\u0301es dans un cadre clinique tre\u0300s strict ; l\u2019auto-me\u0301dication avec ce type de produits est formellement de\u0301conseille\u0301e.<\/p>\n<p><strong>Pour plus d&rsquo;informations et d&rsquo;analyses sur la <a href=\"https:\/\/www.africa-press.net\/sao-tome-e-principe\">S\u00e3o Tom\u00e9 e Pr\u00edncipe<\/a>, suivez <a href=\"https:\/\/www.africa-press.net\/\">Africa-Press<\/a><\/strong><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Africa-Press &#8211; S\u00e3o Tom\u00e9 e Pr\u00edncipe. Un psyche\u0301de\u0301lique issu du venin d\u2019un crapaud toxique pourrait e\u0302tre un traitement contre la de\u0301pression et l\u2019anxie\u0301te\u0301. Ce n\u2019est pas la premie\u0300re fois que la recherche s\u2019inte\u0301resse aux possibilite\u0301s qu\u2019offrent les psyche\u0301de\u0301liques dans le traitement de maladies mentales. Pour le moment, la majorite\u0301 des travaux portait sur un re\u0301cepteur [&hellip;]<\/p>\n","protected":false},"author":82,"featured_media":13365,"comment_status":"open","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[22,10],"tags":[36,55,56],"class_list":["post-13366","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-divers","category-toutes-les-actualites","tag-africa-press","tag-africa-press-sao-tome-e-principe","tag-sao-tome-e-principe"],"yoast_head":"<!-- This site is optimized with the Yoast SEO Premium plugin v26.1 (Yoast SEO v27.0) - https:\/\/yoast.com\/product\/yoast-seo-premium-wordpress\/ -->\n<title>D\u00e9pression : la piste d\u2019un traitement aux toxines hallucinog\u00e8nes de crapaud - S\u00e3o Tom\u00e9 e Pr\u00edncipe<\/title>\n<meta name=\"description\" content=\"Un psyche\u0301de\u0301lique issu du venin d\u2019un crapaud toxique pourrait e\u0302tre un 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